Search results for "Amphiphilic polymer"

showing 3 items of 3 documents

PHEA-PLA biocompatible nanoparticles by technique of solvent evaporation from multiple emulsions

2015

Nanocarriers of amphiphilic polymeric materials represent versatile delivery systems for poorly water soluble drugs. In this work the technique of solvent evaporation from multiple emulsions was applied to produce nanovectors based on new amphiphilic copolymer, the α,β-poly(N-2-hydroxyethyl)-DL-aspartamide-polylactic acid (PHEA-PLA), purposely synthesized to be used in the controlled release of active molecules poorly soluble in water. To this aim an amphiphilic derivative of PHEA, a hydrophilic polymer, was synthesized by derivatization of the polymeric backbone with hydrophobic grafts of polylactic acid (PLA). The achieved copolymer was thus used to produce nanoparticles loaded with α toc…

3003Biocompatible polymerPolymersChemistry PharmaceuticalDrug CompoundingPolyestersalpha-TocopherolPharmaceutical Sciencechemistry.chemical_compoundDrug Delivery SystemsNanoparticlePolylactic acidAmphiphileOrganic chemistryLactic AcidSolubilityDrug CarriersUltrasonic energyPHEA-PLAEmulsionAmphiphilic polymerControlled releaseSolventDrug LiberationSolubilitychemistryChemical engineeringDelayed-Action PreparationsDrug deliveryDrug deliverySolventsNanoparticlesEmulsionsNanocarriersPeptidesDrug carrierHydrophobic and Hydrophilic Interactions
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Cellular Uptake of DNA Block Copolymer Micelles with Different Shapes

2008

The cellular uptake of DNA block copolymer micelles composed of DNA-b-PPO in Caco-2 cells was studied. In particular it was investigated if the shape of micelle aggregates influences the internalization. Rod-like polymeric particles were taken up 12 times more efficiently than their spherical counter parts although they were composed of the same constituents. Furthermore, it was observed that internalization of all the micelle systems was more efficient than the pristine DNA controls. A cytotoxicity assay proved the non-toxic nature of DNA-b-PPO micelle aggregates.

Polymers and PlasticsmicellesOligonucleotidemedia_common.quotation_subjectOrganic Chemistrycellular uptakeNanoparticleCaco-2DNAMicellechemistry.chemical_compoundchemistryCritical micelle concentrationMaterials ChemistryBiophysicsCopolymerOrganic chemistrynanoparticlesamphiphilic polymerInternalizationDrug carrierhybridizationDNAmedia_commonMacromolecular Rapid Communications
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Development and In Vitro Evaluation of Lyotropic Liquid Crystals for the Controlled Release of Dexamethasone.

2017

Made available in DSpace on 2018-12-11T17:33:26Z (GMT). No. of bitstreams: 0 Previous issue date: 2017-08-02 Coordenação de Aperfeiçoamento de Pessoal de Nível Superior (CAPES) In this study, amphiphilic polymers were investigated as biomaterials that can control dexamethasone (DXM) release. Such materials present interfacial properties in the presence of water and an oily phase that can result in lyotropic liquid crystalline systems (LLCS). In addition, they can form colloidal nanostructures similar to those in living organisms, such as bilayers and hexagonal and cubic phases, which can be exploited to solubilize lipophilic drugs to sustain their release and enhance bioavailability. It was…

Materials sciencePolymers and PlasticsAmphiphilic polymersdexamethasone02 engineering and technology030226 pharmacology & pharmacyArticleDexamethasonelcsh:QD241-44103 medical and health scienceschemistry.chemical_compound0302 clinical medicinelcsh:Organic chemistryLyotropicControlled releaseNanostructured systemsLamellar structurelyotropic liquid crystalsIsopropyl myristatedrug releasechemistry.chemical_classificationPolarized light microscopyChromatographySmall-angle X-ray scatteringfungiDrug releaseGeneral ChemistryPolymerkinetic modelKinetic modelamphiphilic polymers; lyotropic liquid crystals; controlled release; drug release; kinetic model; dexamethasone; nanostructured systems021001 nanoscience & nanotechnologyControlled releaseLyotropic liquid crystalschemistryChemical engineeringnanostructured systemsLyotropic liquid crystal0210 nano-technologycontrolled releaseamphiphilic polymersPolymers
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